- Serabelisib - - TAK-117, INK-1117, MLN-1117
- Glesatinib - 格来替尼 - MGCD265
- Emibetuzumab - 依玛妥珠单抗 - LY2875358
- SKB264 - - SKB264
- BT1718 - - BT1718
- EMB01 - - EMB01
- NVL-655 - - NVL-655
- BBT-176 - - BBT-176
- Elzovantinib - - TPX-0022
- Afatinib普来润 - 阿法替尼 - 普来润
- NUV-655 - - NUV-655
- Divarasib - - GDC-6036
- Zotizalkib - - TPX-0131
- Limertinib - - ASK-120067
- Telisotuzumab Vedotin - 特立妥珠单抗 - ABBV-399
- TQB3804 - - TQB3804
- BL-B01D1 - - BL-B01D1
- Taletrectinib - 他雷替尼 - DS-6051b / AB-106
- ZG006 - - ZG006
- TQ-B3139 - - TQ-B3139
- DAJH-1050766 - - DAJH-1050766
- QLH11811 - - QLH11811
- AZD9592 - - AZD9592
- 伊瑞可Gefitinib - 吉非替尼 - 伊瑞可
- Datopotamab - - DS-1062a